Integrin beta-1
Also known as: FNRB, ITGB1, MDF2, MSK12
Function
Integrins alpha-1/beta-1, alpha-2/beta-1, alpha-10/beta-1 and alpha-11/beta-1 are receptors for collagen. Integrins alpha-1/beta-1 and alpha-2/beta-2 recognize the proline-hydroxylated sequence G-F-P-G-E-R in collagen. Integrins alpha-2/beta-1, alpha-3/beta-1, alpha-4/beta-1, alpha-5/beta-1, alpha-8/beta-1, alpha-10/beta-1, alpha-11/beta-1 and alpha-V/beta-1 are receptors for fibronectin. Alpha-4/beta-1 recognizes one or more domains within the alternatively spliced CS-1 and CS-5 regions of fibronectin. Integrin alpha-5/beta-1 is a receptor for fibrinogen. Integrin alpha-1/beta-1, alpha-2/beta-1, alpha-6/beta-1 and alpha-7/beta-1 are receptors for lamimin. Integrin alpha-6/beta-1 (ITGA6:ITGB1) is present in oocytes and is involved in sperm-egg fusion (By similarity). Integrin alpha-4/beta-1 is a receptor for VCAM1. It recognizes the sequence Q-I-D-S in VCAM1. Integrin alpha-9/beta-1 is a receptor for VCAM1, cytotactin and osteopontin. It recognizes the sequence A-E-I-D-G-I-E-L in cytotactin. Integrin alpha-3/beta-1 is a receptor for epiligrin, thrombospondin and CSPG4. Alpha-3/beta-1 may mediate with LGALS3 the stimulation by CSPG4 of endothelial cells migration. Integrin alpha-V/beta-1 is a receptor for vitronectin. Beta-1 integrins recognize the sequence R-G-D in a wide array of ligands. When associated with alpha-7 integrin, regulates cell adhesion and laminin matrix deposition. Involved in promoting endothelial cell motility and angiogenesis. Involved in osteoblast compaction through the fibronectin fibrillogenesis cell-mediated matrix assembly process and the formation of mineralized bone nodules. May be involved in up-regulation of the activity of kinases such as PKC via binding to KRT1. Together with KRT1 and RACK1, serves as a platform for SRC activation or inactivation. Plays a mechanistic adhesive role during telophase, required for the successful completion of cytokinesis. Integrin alpha-3/beta-1 provides a docking site for FAP (seprase) at invadopodia plasma membranes in a collagen-dependent manner and hence may participate in the adhesion, formation of invadopodia and matrix degradation processes, promoting cell invasion. ITGA4:ITGB1 binds to fractalkine (CX3CL1) and may act as its coreceptor in CX3CR1-dependent fractalkine signaling. ITGA4:ITGB1 and ITGA5:ITGB1 bind to PLA2G2A via a site (site 2) which is distinct from the classical ligand-binding site (site 1) and this induces integrin conformational changes and enhanced ligand binding to site 1. ITGA5:ITGB1 acts as a receptor for fibrillin-1 (FBN1) and mediates R-G-D-dependent cell adhesion to FBN1. ITGA5:ITGB1 acts as a receptor for fibronectin FN1 and mediates R-G-D-dependent cell adhesion to FN1. ITGA5:ITGB1 is a receptor for IL1B and binding is essential for IL1B signaling. ITGA5:ITGB3 is a receptor for soluble CD40LG and is required for CD40/CD40LG signaling. Plays an important role in myoblast differentiation and fusion during skeletal myogenesis (By similarity). ITGA9:ITGB1 may play a crucial role in SVEP1/polydom-mediated myoblast cell adhesion (By similarity). Integrins ITGA9:ITGB1 and ITGA4:ITGB1 repress PRKCA-mediated L-type voltage-gated channel Ca(2+) influx and ROCK-mediated calcium sensitivity in vascular smooth muscle cells via their interaction with SVEP1, thereby inhibit vasocontraction.
Classification
- Family (Pfam)
- PF07974 EGF_2, PF23105 EGF_integrin, PF18372 I-EGF_1, PF08725 Integrin_b_cyt, PF07965 Integrin_B_tail, PF00362 Integrin_beta, PF17205 PSI_integrin
- InterPro
- EGF_extracell, EGF_integrin_1, EGF_integrin_2, Integrin_beta_N, Integrin_bsu, Integrin_bsu_cyt_dom, Integrin_bsu_tail, Integrin_bsu_tail_dom_sf, Integrin_bsu_VWA, Integrin_dom_sf, Integrin_I-EGF_CS, PSI, vWFA_dom_sf
- Functional cluster
- Venom Serine Proteases & Phospholipase A2
Experimental structures · PDB · 21
- 3G9W X-ray 2.16A
- 3T9K X-ray 2.30A
- 3VI3 X-ray 2.90A
- 3VI4 X-ray 2.90A
- 4DX9 X-ray 3.00A
- 4WJK X-ray 1.85A
- 4WK0 X-ray 1.78A
- 4WK2 X-ray 2.50A
- 4WK4 X-ray 2.50A
- 7CEB X-ray 2.89A
- 7CEC EM 3.90A
- 7NWL EM 3.10A
- … and 9 more
A predicted model is available from AlphaFold.
Gene Ontology · 106
- GO:0009986 cell surface
- GO:0150053 cerebellar climbing fiber to Purkinje cell synapse
- GO:0032154 cleavage furrow
- GO:0005737 cytoplasm
- GO:0043197 dendritic spine
- GO:0010008 endosome membrane
- GO:0009897 external side of plasma membrane
- GO:0070062 extracellular exosome
- GO:0030175 filopodium
- GO:0005925 focal adhesion
- GO:0097386 glial cell projection
- GO:0034665 integrin alpha1-beta1 complex
- GO:0034680 integrin alpha10-beta1 complex
- GO:0034681 integrin alpha11-beta1 complex
- GO:0034666 integrin alpha2-beta1 complex
- GO:0034667 integrin alpha3-beta1 complex
- GO:0034668 integrin alpha4-beta1 complex
- GO:0034674 integrin alpha5-beta1 complex
- GO:0034677 integrin alpha7-beta1 complex
- GO:0034678 integrin alpha8-beta1 complex
- GO:0034679 integrin alpha9-beta1 complex
- GO:0008305 integrin complex
- GO:0014704 intercalated disc
- GO:0030027 lamellipodium
- GO:0042470 melanosome
- GO:0016020 membrane
- GO:0045121 membrane raft
- GO:0035748 myelin sheath abaxonal region
- GO:0031594 neuromuscular junction
- GO:0048471 perinuclear region of cytoplasm
- GO:0005886 plasma membrane
- GO:0043235 receptor complex
- GO:0055037 recycling endosome
- GO:0001726 ruffle
- GO:0032587 ruffle membrane
- GO:0042383 sarcolemma
- GO:0098685 Schaffer collateral - CA1 synapse
- GO:0045202 synapse
- GO:0097060 synaptic membrane
- GO:0003779 actin binding
- GO:0045296 cadherin binding
- GO:0005509 calcium ion binding
- GO:0050839 cell adhesion molecule binding
- GO:0004895 cell adhesion receptor activity
- GO:0098639 collagen binding involved in cell-matrix adhesion
- GO:0015026 coreceptor activity
- GO:0001968 fibronectin binding
- GO:0005178 integrin binding
- GO:0098640 integrin binding involved in cell-matrix adhesion
- GO:0043236 laminin binding
- GO:0000287 magnesium ion binding
- GO:0002020 protease binding
- GO:0046982 protein heterodimerization activity
- GO:0019901 protein kinase binding
- GO:1990782 protein tyrosine kinase binding
- GO:0044877 protein-containing complex binding
- GO:0001618 virus receptor activity
- GO:0001525 angiogenesis
- GO:0030183 B cell differentiation
- GO:0071711 basement membrane organization
- GO:0007161 calcium-independent cell-matrix adhesion
- GO:0023035 CD40 signaling pathway
- GO:0007155 cell adhesion
- GO:0033627 cell adhesion mediated by integrin
- GO:0016477 cell migration
- GO:0030030 cell projection organization
- GO:0098609 cell-cell adhesion
- GO:0033631 cell-cell adhesion mediated by integrin
- GO:0007160 cell-matrix adhesion
- GO:0031589 cell-substrate adhesion
- GO:0006968 cellular defense response
- GO:0071404 cellular response to low-density lipoprotein particle stimulus
- GO:0000132 establishment of mitotic spindle orientation
- GO:0030198 extracellular matrix organization
- GO:0034113 heterotypic cell-cell adhesion
- GO:0007156 homophilic cell-cell adhesion
- GO:0007229 integrin-mediated signaling pathway
- GO:0030032 lamellipodium assembly
- GO:0007159 leukocyte cell-cell adhesion
- GO:0050901 leukocyte tethering or rolling
- GO:0035633 maintenance of blood-brain barrier
- GO:0048333 mesodermal cell differentiation
- GO:0007517 muscle organ development
- GO:0045445 myoblast differentiation
- GO:0007520 myoblast fusion
- GO:2000811 negative regulation of anoikis
- GO:0045906 negative regulation of vasoconstriction
- GO:0006909 phagocytosis
- GO:0045766 positive regulation of angiogenesis
- GO:0043065 positive regulation of apoptotic process
- GO:0030335 positive regulation of cell migration
- GO:0045743 positive regulation of fibroblast growth factor receptor signaling pathway
- GO:0010763 positive regulation of fibroblast migration
- GO:0051951 positive regulation of glutamate uptake involved in transmission of nerve impulse
- GO:0043547 positive regulation of GTPase activity
- GO:0051897 positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction
- GO:1903078 positive regulation of protein localization to plasma membrane
- GO:1900748 positive regulation of vascular endothelial growth factor signaling pathway
- GO:0090303 positive regulation of wound healing
- GO:0150103 reactive gliosis
- GO:0031623 receptor internalization
- GO:0010710 regulation of collagen catabolic process
- GO:0150003 regulation of spontaneous synaptic transmission
- GO:1905806 regulation of synapse pruning
- GO:0014850 response to muscle activity
- GO:0035313 wound healing, spreading of epidermal cells
Drugs targeting this protein · 2
- FIRATEGRAST antagonist
- ATN-161 antagonist
Related proteins · sequence + function similarity
- Integrin beta-1 1.00
- Integrin beta-1 1.00
- Integrin beta-1 1.00
- Integrin beta-1 1.00
- Integrin beta-1 1.00
- Integrin beta-1 0.99
- Integrin beta-1 0.99
- Integrin beta-1 0.99
- Integrin beta-1 0.98
- Integrin beta-1-B 0.98
- Integrin beta-1-A 0.98
- Integrin beta pat-3 0.93
Co-cited proteins · studied together in the literature
- Integrin alpha-5 16 shared papers
- Arf-GAP with coiled-coil, ANK repeat and PH domain-containing protein 1 2 shared papers
- Integrin beta-1-binding protein 1 5 shared papers
- Integrin alpha-4 8 shared papers
- Integrin alpha-2 4 shared papers
- Neisseria adhesin A 1 shared papers
- Nicotinamide riboside kinase 2 1 shared papers
- Fermitin family homolog 2 2 shared papers
- Integrin beta-1 8 shared papers
- Glycoprotein 1 shared papers
- Protein BMRF2 1 shared papers
- Integrin alpha-V 11 shared papers
Literature · 79 cited papers
- The C-type lectin domain of CD62P (P-selectin) functions as an integrin ligand. Life. Sci Alliance · 2023
- The integrin ligand SVEP1 regulates GPCR-mediated vasoconstriction via integrins alpha9beta1 and alpha4beta1. Br. J. Pharmacol. · 2022
- PEAK1 Y635 phosphorylation regulates cell migration through association with Tensin3 and integrins. J. Cell Biol. · 2022
- Structural insights into integrin alpha5beta1 opening by fibronectin ligand. Sci. Adv. · 2021
- The Integrin Binding Peptide, ATN-161, as a Novel Therapy for SARS-CoV-2 Infection. JACC Basic Transl. Sci. · 2021
- GRP78 and Integrins Play Different Roles in Host Cell Invasion during Mucormycosis. MBio · 2020
- Integrin beta1 Promotes Peripheral Entry by Rabies Virus. J. Virol. · 2020
- Integrin Binding to the Trimeric Interface of CD40L Plays a Critical Role in CD40/CD40L Signaling. J. Immunol. · 2019
- Direct binding to integrins and loss of disulfide linkage in interleukin-1beta (IL-1beta) are involved in the agonistic action of IL-1beta. J. Biol. Chem. · 2017
- N-terminome analysis of the human mitochondrial proteome. Proteomics · 2015
- Proinflammatory secreted phospholipase A2 type IIA (sPLA-IIA) induces integrin activation through direct binding to a newly identified binding site (site 2) in integrins alphavbeta3, alpha4beta1, and alpha5beta1. J. Biol. Chem. · 2015
- Mapping of SUMO sites and analysis of SUMOylation changes induced by external stimuli. Proc. Natl. Acad. Sci. U.S.A. · 2014
- … and 67 more in the literature graph